松香马来酸酐衍生物的制备及生物活性  

Synthesis and Biological Activity of Maleopimaric Acid Derivatives

作　　者：王恒山[1] 谢建武[1] 潘英明[1] 黎霜 苏桂发[1] 文进军[1] 

机构地区：[1]广西师范大学化学化工学院,桂林541004 [2]桂林市药检所,桂林541004

出　　处：《农药》2005年第11期506-508,共3页Agrochemicals

基　　金：国家自然科学基金(No.20362002);广西青年科学基金(No.0229023);广西高校百名中青年学科带头人资助计划资助项目

摘　　要：合成了3类共5种松香马来酸酐衍生物,并进行了结构表征。生物活性测定结果表明化合物2a、2b和2c均具有植物激素作用。化合物2a～2c的合成采用无溶剂绿色化学的合成方法,合成反应操作简便,产率达90%,适合规模化生产。Five of three series maleopimaric acid derivatives are synthesized. The biological tests indicate that compounds 2a, 2b and 2c exhibite remarkable plant hormone activities. Compounds 2a-2c are synthesized through solvent free green chemistry reaction which can be finished very quickly with high yield （over 90%）, the work-up is simple, so the derivatives can be produced in large-scale.

关 键 词：松香 松香马来酸酐 取代苯脲 酰腙 酰胺基硫脲 

分 类 号：TQ450.1[化学工程—农药化工]