N-[5-(1-邻氯苯氧乙基)-1,3,4-噻二唑-2-基]-N′-芳氧乙酰基硫脲的合成与生物活性  

Synthesis and Biological Activity of N-[5-(1-o-Chlorophenoxyethyl)-1,3,4-thiodiazol-2-yl]- N′-aryloxyacetyl Thioureas

作　　者：王子云[1] 王胜[2] 宋新建[2] 汪焱钢[2] 

机构地区：[1]周口师范学院化学系,河南周口466000 [2]华中师范大学化学学院,湖北武汉430079

出　　处：《农药学学报》2005年第3期282-284,共3页Chinese Journal of Pesticide Science

基　　金：国家自然科学基金(20072009)资助项目

摘　　要：为了寻找新的高生物活性农药,通过2-氨基-5-(1-邻氯苯氧乙基)-1,3,4-噻二唑与芳氧乙酰基异硫氰酸酯反应,合成了9个新的芳氧乙酰基硫脲,初步的生物活性测定结果表明,部分目标化合物具有良好的植物生长调节活性,其中2 c、2d具有较好的生长素活性,其生长促进率分别为26.9%和27.2%。In order to search for high biological active pesticide, nine novel aryloxyacetyl thioureas have been synthesized by the reaction of 2-amino-5-（1-o-chlorophenoxyethyl）-1,3,4-thiodiazole with aryloxyacetyl isothiocyanates. The preliminary biological activity tests exhibited that some target compounds possessed a good activity as plant growth regulator, and 2c and 2d had better activities as auxin, the oromoting rate were 26.9% and 27.9%.

关 键 词：酰基硫脲 1 3 4-噻二唑 合成 生物活性 生长素 

分 类 号：O626.27[理学—有机化学]