1-芳基-5-吡唑酰胺类化合物的合成与生物活性研究  

Synthesis and Biological Activity of Novel 1-Phenyl-5-pyrazolecarboxamide Derivatives

作　　者：郭丽琴[1] 徐尚成[1] 马海军[1] 倪珏萍[1] 侯华民[1] 刘丽[1] 万琴[1] 

机构地区：[1]江苏省农药研究所股份有限公司,南京210019

出　　处：《农药研究与应用》2008年第2期15-18,共4页Agrochemicals Research & Application

摘　　要：本文充分考虑取代吡唑类农药品种吡螨胺(MK-239)和氟虫腈的结构特点与异同之处,设计合成了18个1-芳基-5-吡唑酰胺类新化合物,并通过核磁进行了结构表征。初步生物活性测定表明部分化合物表现出优良的杀虫杀菌活性。Eighteen novel N-phenyl-3-pyrazolecarboxamide derivatives were designed and synthesized through combining the structural characteristics of commercially pesticides MK-239 and Regent. These compounds were confirmed by ~H NMR. The preliminary bioassay showed that some of them exhibited good insecticidal and germicidal activities.

关 键 词：1-芳基-5-吡唑酰胺 合成 生物活性 

分 类 号：O621.3[理学—有机化学]