中乌头碱结构中磺酰基的引入及其杀虫活性的测定  

Sulfoacylation of Mesaconitine and Its Insecticidal Activity

作　　者：王惠[1] 侯大斌[1] 杨海君[1] 袁小红[1] 许源[1] 赵祥升[1] 

机构地区：[1]西南科技大学生命科学与工程学院,四川绵阳621010

出　　处：《湖北农业科学》2009年第3期718-720,共3页Hubei Agricultural Sciences

基　　金：国家"十一五"科技支撑计划重大专项课题(2006BAE01A01-12)

摘　　要：通过化学方法向中乌头碱结构中引入磺酰基,对产物进行杀虫活性的测定。发现甲磺酰化与苯磺酰化中乌头碱对苜蓿蚜(Aphis medicagini)的杀虫活性72h之内达到50%,较中乌头碱杀虫活性提高了20%。The sulfonyl compound of mesaconitine was prepared and its insecticidal activity was studied in this paper. The results revealed that the insecticidal activity of methane sulfonyl compound and benzene sulfonyl compound to Aphis medicagini could reach 50% in 72 h which was 20% higher than that by mesaconitine.

关 键 词：中乌头碱 磺酰化 杀虫活性 

分 类 号：R284.3[医药卫生—中药学]