Selective mono-arylation in palladium-catalyzed cross-coupling reaction of dichlorotriazines with phenylboronate ester derivatives  

作　　者：Jin-Fu Dong Xin Yu Cheng-Qing Ning Liang Hu Nie-Fang Yu 

机构地区：[1]School of Pharmaceutical Sciences,Central South University [2]School of Pharmaceutical Sciences,Sun Yat-sen University

出　　处：《Chinese Chemical Letters》2013年第1期41-44,共4页中国化学快报（英文版）

基　　金：the National Natural Science Foundation of China(Nos.30873137,30772645 and 81172927) for their financial support

摘　　要：Palladium-catalyzed cross-coupling reaction between dichlorotriazines and phenylboronate esters produced the mono-awlated triazines selectively and thus, the corresponding phenyltriazine derivatives could be assembled efficiently in moderate to good overall yields （50-80%）.Palladium-catalyzed cross-coupling reaction between dichlorotriazines and phenylboronate esters produced the mono-awlated triazines selectively and thus, the corresponding phenyltriazine derivatives could be assembled efficiently in moderate to good overall yields （50-80%）.

关 键 词：Suzuki cross-coupling reactionDichlorotriazinesAryl boronic estersPd（PPh3）4 

分 类 号：O643.32[理学—物理化学]