啶酰菌胺合成方法的研究进展  

Progress on Synthesis of Boscalid

作　　者：朱思佳 刘明成[1] 杨建华 宋华月 王洋洋 刘雷芳[1] ZHU Si-jia;LIU Ming-cheng;YANG Jian-hua;SONG Hua-yue;WANG Yang-yang;LIU Lei-fang(Key Laboratory of Coordination Chemistry and Functional Materials in Universities of Shandong, Dezhou University, Dezhou 253023, China;Chemical Teaching and Research Group, Dezhou No. 1 Middle School, Dezhou 253023, China)

机构地区：[1]德州学院山东高校配位化学与功能材料重点实验室,山东德州253023 [2]山东省德州市第一中学化学教研组,山东德州253023

出　　处：《化学试剂》2018年第7期647-652,共6页Chemical Reagents

基　　金：山东省自然科学基金资助项目(ZR2014BL009、ZR2014BL001);国家大学生创新创业训练计划项目(201510448061);国家星火计划项目(2015GA740090)

摘　　要：作为一种广谱、低毒、高效的新型杀菌剂,啶酰菌胺引起了国内外的广泛关注,研究、开发和改进现有啶酰菌胺的工业生产路线势在必行,这不但能提升我国农药生产企业的核心竞争力,而且还将给农业增收、农药市场带来巨大的发展机遇。到目前为止,文献中报道了较多啶酰菌胺的合成方法。为了更好的把握啶酰菌胺的合成现状,根据原料的不同,从氯代芳烃、碘代芳烃、溴代芳烃和其他原料4个角度对啶酰菌胺的合成路线进行了综述,以期对同行工作者有所启发和帮助。Boscalid,a new and important fungicide,has attracted wide attention both at home and abroad due to its broad spectrum,low toxicity and high efficiency.It is very necessary to study,explore,and improve the existing synthetic route of Boscalid,which are very important not only for the competitive power of pesticide production enterprises but also for agriculture incomes and the development of pesticide market.There have been many synthetic methods in literature.This work,which should be helpful for the researchers of Boscalid,reviewed the synthetic methods for Boscalid in literature.Based on the raw materials used,this work is organized in the sequence of aryl chlorides,aryl iodides,aryl bromides and other materials.

关 键 词：啶酰菌胺 合成 研究进展 

分 类 号：O625.13[理学—有机化学]