氟吡呋喃酮及其类似物研究进展  

Recent research progress on flupyradifurone and its analogues

作　　者：苏彦豪 许磊川 赵宇[1] 张倩[1] 李益豪 王明安[1] SU Yanhao;XU Leichuan;ZHAO Yu;ZHANG Qian;LI Yihao;WANG Ming’an(Innovation Center of Pesticide Research,Department of Applied Chemistry,China Agricultural University,Beijing 100193,China)

机构地区：[1]中国农业大学应用化学系,农药创新研究中心,北京100193

出　　处：《农药学学报》2022年第3期435-451,共17页Chinese Journal of Pesticide Science

基　　金：国家自然科学基金(21772229).

摘　　要：氟吡呋喃酮(flupyradifurone)是拜耳公司开发的新型丁烯内酯类杀虫剂,对刺吸式口器害虫具有优异的杀虫活性,与现有商品化新烟碱类杀虫剂相比,其作用机制独特,对蜜蜂低毒,自2014年上市以来就成为了农药学研究领域的热点。本文从氟吡呋喃酮的创制过程、生物活性及抗性、作用机制、代谢残留、对蜜蜂等非靶标生物的影响以及结构修饰等方面对该产品进行了综述。Flupyradifurone,a new butenolide insecticide developed by Bayer Cropscience AG,has excellent insecticidal activity against sucking pests.Compared with the existing commercial neonicotinoid insecticides,it has a unique mode of action and is low toxicity to bees.Therefore,it has been one of the hot research topics in the agrochemical field since it was launched in 2014.The creation process,bioactivity and resistance,mechanism of action,metabolic residue,effects on non-target organisms such as bees and structural modification of fluopyradifurone were summarized in this review.

关 键 词：氟吡呋喃酮 丁烯内酯 生物活性 结构改造 综述 

分 类 号：TQ453.2[化学工程—农药化工]