Modelling One-Pot Method for Synthesis of 2,3-Dihydro-1<i>H</i>-pyrrolo[2,1-<i>c</i>][1,4]benzothiazine 5,5-Dioxides and Their Homologues  

作　　者：Oleksandr Yu Grevtsov Oleg V. Zaremba Anna B. Bondarenko Oleksandr G. Drushlyak Sergiy M. Kovalenko Valentyn P. Chernykh 

机构地区：[1]National University of Pharmacy, Kharkiv, Ukraine

出　　处：《International Journal of Organic Chemistry》2013年第2期125-135,共11页有机化学国际期刊（英文）

摘　　要：A facile method for synthesis of 2,3-dihydro-1H-pyrrolo[2,1-c][1,4]benzothiazines by interaction of methylenactive (2-fluorophenyl)sulfones with homologues of either 5-methoxy-3,4-dihydro-2H-pyrrole or 5-(methylthio)-3,4-dihydro- 2H-pyrrole has been developed.A facile method for synthesis of 2,3-dihydro-1H-pyrrolo[2,1-c][1,4]benzothiazines by interaction of methylenactive (2-fluorophenyl)sulfones with homologues of either 5-methoxy-3,4-dihydro-2H-pyrrole or 5-(methylthio)-3,4-dihydro- 2H-pyrrole has been developed.

关 键 词：SULFONES Lactims Cyclization Heterocycles Nucleophilic Aromatic Substitution 

分 类 号：O6[理学—化学]