supported by the National Key R&D Program of China (2022YFA1506100);the National Natural Science Foundation of China (21901191);the Fundamental Research Funds for the Central Universities (2042023kf0202);the China Postdoctoral Science Foundation (2023TQ0250)。
Previous carbene insertion to C–H bonds of 1,3-azoles relied on metal carbene species. Herein, we report a metal-free C(sp^(2))–H bond functionalization of 1,3-azoles with trifluoroacetylsilanes. The reaction featur...
partially supported by National Natural Science Foundation of China [21172181, 81250110089, 81250110554 (The Research Fellowship for International Young Scientists from International (Regional) Cooperation and Exchange Program)];the key program from Natural Science Foundation of Chongqing (CSTC2012jjB10026);the Specialized Research Fund for the Doctoral Program of Higher Education of China (SRFDP 20110182110007);the Fundamental Research Funds for the Central Universities (the key program XDJK2012B026)
A series of naphthalimide azoles as potential antibacterial and antifungal agents were conveniently and efficiently synthesized starting from commercially available 6-bromobenzo[de]isochromene-l,3-dione. All the new c...