Fe(OTf)_(3) Catalyzed Annulation of 2,3-Disubstituted Indoles with Aziridines  

作　　者：Hua Liu Chao Zheng Shu-Li You 

机构地区：[1]State Key Laboratory of Organometallic Chemistry,Shanghai Institute of Organic Chemistry,Chinese Academy of Sciences,Shanghai 200032,China

出　　处：《Chinese Journal of Chemistry》2014年第8期709-714,共6页中国化学（英文版）

基　　金：We thank the National Basic Research Program of China(No.2010CB833300);the National Natural Science Foundation of China(Nos.21025209,21121062,21332009,and 21302209)for generous financial support.

摘　　要：A Fe(OTf)_(3) catalyzed[3+2]annulation reaction between 2,3-disubstituted indoles and N-Ts aziridines is described herein.A series of hexahydropyrrolo[3,4-b]indole derivatives bearing two consecutive quaternary carboncenters can be generated efficiently.The reaction features cheap catalyst,mild conditions and operational simplicity.

关 键 词：ANNULATION INDOLE AZIRIDINE Lewis acid catalysis 

分 类 号：O62[理学—有机化学]