Soluble Polymer-supported Synthesis of Indoles via Palladium-mediat-ed Heteroannulation of Terminal Alkynes with o-Iodoanilines  

作　　者：Xu Feng LIN Cheng MA Ye Wei YANG Yan Guang WANG 

机构地区：[1]Department of Chemistry,Zhejiang University,Hangzhou 310027

出　　处：《Chinese Chemical Letters》2002年第8期705-707,共3页中国化学快报(英文版)

基　　金：the National Natural Science Foundation of China (No. 29972037) and Foundation for University Key Teacher by the Ministry of Education.

摘　　要：A soluble polymer-supported synthesis of indoles via palladium-mediated hetero- annulation of terminal alkynes with o-iodoanilines has been described. The protocol provides a useful tool for constructing combinatorial indole libraries.A soluble polymer-supported synthesis of indoles via palladium-mediated hetero- annulation of terminal alkynes with o-iodoanilines has been described. The protocol provides a useful tool for constructing combinatorial indole libraries.

关 键 词：INDOLE polyethylene glycol(PEG) liquid-phase. 

分 类 号：O633[理学—高分子化学]