PHOSPHODIESTERASE

作品数:80被引量:149H指数:6
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相关领域:医药卫生更多>>
相关作者:朱永通徐雯曹云燕崔倩倩蔡圣朝更多>>
相关机构:南方医科大学南方医院浙江大学安徽中医药大学华中农业大学更多>>
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相关基金:国家自然科学基金国家重点基础研究发展计划国家科技支撑计划北京市自然科学基金更多>>
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Discovery of a highly specific ^(18)F-labeled PET ligand for phosphodiesterase 10A enabled by novel spirocyclic iodonium ylide radiofluorination
《Acta Pharmaceutica Sinica B》2022年第4期1963-1975,共13页Zhiwei Xiao Huiyi Wei Yi Xu Ahmed Haider Junjie Wei Shiyu Yuan Jian Rong Chunyu Zhao Guocong Li Weibin Zhang Huangcan Chen Yuefeng Li Lingling Zhang Jiyun Sun Shaojuan Zhang Hai-Bin Luo Sen Yan Qijun Cai Lu Hou Chao Che Steven H.Liang Lu Wang 
the support of K.C.Wong Education Foundation (China);financially supported by the National Natural Science Foundation of China (No.82071974);Shenzhen Basic Research Project (JCYJ20180503182116931, China);Guangdong Basic and Applied Basic Research Foundation (2020A1515011192, 2018A0303130052, China);Guangzhou Key Research Program on Brain Science (202007030008, China);the Fundamental Research Funds for the Central Universities (21619104, 21621051, China)
As a member of cyclic nucleotide phosphodiesterase(PDE)enzyme family,PDE10A is in charge of the degradation of cyclic adenosine(cAMP)and guanosine monophosphates(cGMP).While PDE10A is primarily expressed in the medium...
关键词:Phosphodiesterase 10A PET radioligand 18F Spirocyclic iodonium ylide Nonhuman primate Target occupancy 
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