云南高校图书馆联盟文献共享服务平台- PYRAZOL

PYRAZOL: 作品数：93被引量：65H指数：4; 导出分析报告; 相关领域：理学更多>>; 相关作者：温国山曾裕平李峰胡春李大伟更多>>; 相关机构：安阳师范学院中国医药大学静宜大学商丘师范学院更多>>; 相关期刊：《Chinese Physics Letters》《Journal of Chemistry and Chemical Engineering》《Chinese Journal of Structural Chemistry》《Journal of Materials Science and Chemical Engineering》更多>>; 相关基金：国家自然科学基金国家重点基础研究发展计划天津市自然科学基金国家教育部博士点基金更多>>

Synthesis, Structural Characterization and Antimicrobial Activity of a Novel Cobalt(II) Complex Based on 3-Methyl-1-Phenyl-4-(2-Thienoyl)-Pyrazol-5-One: 《Journal of Materials Science and Chemical Engineering》2023年第8期109-126,共18页Emeline Sorelle Mefouegang Claudelle Sybilline Anensong Djadock Golngar Djimassingar Gabriel Tchuente Kamsu Donald Raoul Tchuifon Tchuifon Alain Charly Tagne Kuate Dirk Bockfeld Jean Ngoune; New cobalt(II) complex, [Co(O₂C₁₅H₁₁N₂S)₂(OH₂)₂]∙2H₂O (1∙2H₂O), has been synthesized upon reaction of cobalt chloride ...; 关键词：COBALT ACYLPYRAZOLONE X-Ray Diffraction Antimicrobial Activity 3-Methyl-1-Phenyl-4-(2-Thienoyl)-Pyrazol-5-One

Synthesis, Structural Characterization and Antimicrobial Activity of a Novel Cobalt(II) Complex Based on 3-Methyl-1-Phenyl-4-(2-Thienoyl)-Pyrazol-5-One: 《Journal of Modern Physics》2023年第8期109-126,共12页Emeline Sorelle Mefouegang Claudelle Sybilline Anensong Djadock Golngar Djimassingar Gabriel Tchuente Kamsu Donald Raoul Tchuifon Tchuifon Alain Charly Tagne Kuate Dirk Bockfeld Jean Ngoune; New cobalt(II) complex, [Co(O₂C₁₅H₁₁N₂S)₂(OH₂)₂]∙2H₂O (1∙2H₂O), has been synthesized upon reaction of cobalt chloride ...; 关键词：COBALT ACYLPYRAZOLONE X-Ray Diffraction Antimicrobial Activity 3-Methyl-1-Phenyl-4-(2-Thienoyl)-Pyrazol-5-One

Structure-activity relationship of pyrazol-4-ylpyridine derivatives and identification of a radiofluorinated probe for imaging the muscarinic acetylcholine receptor M4: 《Acta Pharmaceutica Sinica B》2023年第1期213-226,共14页Ahmed Haider Xiaoyun Deng Olivia Mastromihalis Stefanie K.Pfister Troels E.Jeppesen Zhiwei Xiao Vi Pham Shaofa Sun Jian Rong Chunyu Zhao Jiahui Chen Yinlong Li Theresa R.Connors April T.Davenport James B.Daunais Vahid Hosseini Wenqing Ran Arthur Christopoulos Lu Wang Celine Valant Steven H.Liang; supported by the Swiss National Science Foundation(SNSF);supported by the National Health and Medical Research Council(NHMRC)Program Grant(APP1055134,USA);the Australian Research Council(ARC)Discovery Project(DP190102950,USA);supported by grants from Fulbright Denmark,The Lundbeck Foundation,Eva and Henry Frònkels foundation,The Danish Cancer Society,The Harboe Foundation。; There is an accumulating body of evidence implicating the muscarinic acetylcholine receptor4(M4)in schizophrenia and dementia with Lewy bodies,however,a clinically validated M4positron emission tomography(PET)radiolig...; 关键词：Muscarinicacetylcholine receptor Positronemission tomography NEUROIMAGING NEUROPHARMACOLOGY Neurological disorders

Catalyst-free ultrasound assisted novel one pot pseudo five component synthesis of aryl-bis-[1H-pyrazol-5-ol-4-yl]methanes,het(aryl)-bis-[1H-pyrazol-5-ol-4-yl]methanes and their 1-phenyl derivatives in aqueous medium: 《Green Synthesis and Catalysis》2022年第2期190-193,共4页Sudha S Mohamed Afzal Pasha; Dr.Mohamed Afzal Pasha acknowledges the University Grants Commission(UGC),New Delhi,INDIA for the BSR Faculty Fellowship(No.F.18–1/2011(BSR),November 2019).; An efficient,catalyst-free and eco-friendly ultrasound-assisted novel one-pot pseudo-five-component synthesis of aryl-bis-[1H-pyrazol-5-ol-4yl]methanes,het(aryl)-bis-[1H-pyrazol-5-ol-4yl]methanes and their 1-phenyl de...; 关键词：Bis pyrozolyl-methanes Ethyl acetoacetate Aromatic/het(aryl)aldehydes Hydrazine/phenyl hydrazine One-pot multi-component synthesis Ultrasound

Discovery of 4-cyclopropyl-3-(2-((1-cyclopropyl-1H-pyrazol-4-yl) amino) quinazolin-6-yl)-N-(3-(trifluoromethyl) phenyl) benzamides as potent discoidin domain receptor inhibitors for the treatment of idiopathic pulmonary fibrosis被引量：1: 《Acta Pharmaceutica Sinica B》2022年第4期1943-1962,共20页Qi Wang Bixi Tang Dandan Sun Ying Dong Yinchun Ji Huanyu Shi Liwei Zhou Yueyue Yang Menglan Luo Qian Tan Lin Chen Yue Dong Cong Li Rongrong Xie Yi Zang Jingkang Shen Bing Xiong Jia Li Danqi Chen; This research has been financially supported by grants from the Strategic Priority Research Program of the Chinese Academy of Sciences(Grant No.XDA12020323);the National Science&Technology Major Project“Key New Drug Creation and Manufacturing Program”of China(Grant No.2018ZX09711002-004-009);the Strategic Priority Research Program of Chinese Academy of Sciences(No.SIMM010203);Institutes for Drug Discovery and Development,Chinese Academy of Sciences(No.CASIMM0120215009);National Natural Science Foundation of China(No.U1703235);Shanghai Science and Technology Development Funds(18431907100,China).; Idiopathic pulmonary fibrosis(IPF)is a chronic fatal lung disease with a median survival time of 3–5 years.Inaccurate diagnosis,limited clinical therapy and high mortality together indicate that the development of ef...; 关键词：Idiopathic pulmonary fibrosis Discoidin domain receptor Kinase Inhibitor Docking

Design, Synthesis, and Evaluation of Fungicidal Activity of Novel Pyrazole-Containing Strobilurin Derivatives被引量：1: 《Chinese Journal of Chemistry》2021年第6期1531-1537,共7页Zesheng Hao Weibo Wang Bin Yu Xin Qi You Lv Xiaoyu Liu Haoyin Chen Tatiana A.Kalinina Tatiana V.Glukhareva Zhijin Fan; the National Natural Science Foundation of China(No.31872007);the Tianjin Natural Science Foundation(No.18JCZDJC33500);the International Science&Technology Cooperation Program of China(No.2014DFR41030);the Tianjin Development Program for Innovation and Entrepreneurship.; In searching for novel fungicidal leads,a series of pyrazole-containing strobilurins were rationally designed,synthesized and charac-terized.Bioassay indicated that compound 1-7 displayed excellent fungicidal activity...; 关键词：Drug design STROBILURINS Biological activity Structure-activity relationships Cytochrome bc_(1)complex

Four Complexes of Mn(Ⅱ),Co(Ⅱ),Ni(Ⅱ)and Cu(Ⅱ)Based on 2-Morpholine-4-yl-4,6-di-pyrazol-1-yl-1,3,5-triazine: 《Chinese Journal of Structural Chemistry》2021年第6期729-738,684,共11页TIAN Wen-Yu CHU Jin-Feng; Three azide bridged complexes,namely,[Mn_(2)L_(2)(N_(3))_(4)(H_(2)O)_(2)](1),[Co_(2)L_(2)(N_(3))_(4)]·(H_(2)O)_(3)(2)and[Ni_(2)L_(2)(N_(3))_(3)(H_(2)O)]N_(3)·(H_(2)O)4(3)(L=2-morpholine-4-yl-4,6-di-pyrazol-1-yl-1,3,...; 关键词：azide bridged complexes supramolecular crystal structure THIOCYANATE

Syntheses, Structures and Photoluminescence of Novel Lanthanide-organic Frameworks Based on 1, 4-Bis(3,5-dicarboxylic pyrazol-1-ylmethyl) Benzene: 《Chinese Journal of Structural Chemistry》2020年第5期960-966,共7页LI Chuang HE Yong-Ke SHAO Na XIONG Gang WU Shuang-Yan YOU Li-Xin SUN Ya-Guang; supported by the National Natural Science Foundation of China(21701116,21671139 and 21501122);the Doctor Scientific Research Foundation of Liaoning Province(201601201 and 201601193);Program for Liaoning Innovative Research Team in University(No.2018012)。; Two isomorphic 3D lanthanide metal-organic frameworks,{[Tb(L)0.5(OX)0.5(H2 O)2DMF]·DMF}n(1)and{[Dy(L)0.5(OX)0.5(H2 O)2 DMF]·DMF}n(2),have been prepared under solvothermal conditions based on l,4-bis(3,5-dicarboxylic...; 关键词：lanthanide-organic frameworks luminescent emission antenna effect

One Novel Tetranuclear Copper Cluster by 2-(1H-Pyrazol-3-yl)pyridine:Synthesis, Structure and Properties: 《Chinese Journal of Structural Chemistry》2020年第5期949-954,共6页ZHU Mei XIE Wei-Nan YANG Mai-E HUA Feng-Zhen ZHANG Guo-Ning WANG Yu-Cheng ZHAO Hong; financially supported by the Jiangsu Ainaji Neoenergy Science&Technology Co.,Ltd.(8507040091);the Fundamental Research Funds for the Central Universities(3207045420);the National Natural Science Foundation of China(81703366)。; A novel tetranuclear copper cluster[Cu4(μ-L)6Cl2]was constructed by 2-(1H-pyrazol-3-yl)pyridine(HL)under hydrothermal conditions,and structurally concluded by single-crystal X-ray diffractions,elemental analyses and ...; 关键词：2-(1H-pyrazol-3-yl)pyridine tetranuclear copper cluster fluorescent property

Synthesis and biological evaluation of a series of2-(((5-akly/aryl-1H-pyrazol-3-yl)methyl)thio)-5-alkyl-6-(cyclohexylmethyl)-pyrimidin-4(3H)-ones as potential HIV-1 inhibitors被引量：3: 《Acta Pharmaceutica Sinica B》2020年第3期512-528,共17页Yumeng Wu Chengrun Tang Ruomei Rui Liumeng Yang Wei Ding Jiangyuan Wang Yiming Li Christopher C.Lai Yueping Wang Ronghua Luo Weilie Xiao Hongbing Zhang Yongtang Zheng Yanping He; Financial support from the National Natural Science Foundation of China(Grant No.U1702286,21262044,81660612,21362017,21762048);Program for Changjiang Scholars and Innovative Research Team in University(IRT_17R94,China);The Key Scientific and Technological Program of China(2017ZX09101004-014-007);The Yunnan Applicative and Basic Research Program(P0120150150,2018FA048,China);Project of Innovative Research Team of Yunnan Province to Weilie Xiao;Shanghai Chem Partner Co.,Ltd.for completing the Pharmacokinetics Assays.; A series of 2-(((5-akly/aryl-1 H-pyrazol-3-yl)methyl)thio)-5-alkyl-6-(cyclohexylmethyl)-pyrimidin-4(3 H)-ones were synthesized and their anti-HIV-1 activities were evaluated.Most of these compounds were highly active ...; 关键词：HIV-1 NNRTIS S-DABOs Antiviral activity SAR Molecular modeling

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