support from the National Natural Science Foundation of China(51802001);Education Committee of Anhui Province(KJ2018A0037).
A transition-metal free three-component coupling reaction of azaindoles,C_(60),and bromoalkanes/triphenylamines has been developed to provide an efficient access to diverse azaindole functionalized 1,4-C_(60) adducts....
A catalyst- and solvent-free protocol for the synthesis of 7-azagramine analogues is described via a three-component Mannich type reaction between 7-azaindole, aromatic aldehydes and heterocyclic amines in acceptable ...
This work was supported by the National Natural Science Foundation of China (51373072, 21262015, 21162011, 21363009), the Project of Jiangxi Advantage Sci-Tech Innovative Team (20142BCB24012), the Science Funds of Natural Science Foundation of Jiangxi Province (20132BAB203005, 20142BAB203005), and the Project of the Science Funds of Jiangxi Education Office (KJLD12035, GJJ12587, GJJ14592).
Three new asymmetrical diarylethenes containing an azaindole moiety and a variable heteroaryl ring have been synthesized. Their properties, such as photochromism, fatigue resistance, thermal stability, acidichromism, ...
We designed and synthesized a 7-azaindole derivative(TH1082), which was characterized by 1^H NMR and 13^C-NMR. We investigated its antitumor effects on human melanoma A375 cells, human liver cancer SMMC cells and hu...
supported by the Shanghai Family Planning Commission Research Fund(No2007JG02);Shanghai Leading Academic Discipline Project(NoB906)
A series of 7-azaindol derivatives were designed based on the homologous 3D model of human acrosin.These compounds were synthesized and evaluated for their human acrosin inhibitory activities in vitro.Compounds 7a,7i,...