2-AMINOTHIAZOLE

作品数：8被引量：15H指数：2
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相关期刊：《Chinese Journal of Chemistry》《Chemical Research in Chinese Universities》《Chinese Chemical Letters》更多>>
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Identification of 2-aminothiazoyl piperidine derivatives as a new class of adjuvants potentiating the activity of colistin against Acinetobacter baumannii
《Chinese Chemical Letters》2023年第2期468-474,共7页Yuce Chen Zhen Li Yu Yin Ping Yang Yijin Kong Zhong Li Daijie Chen Xiaoyong Xu 
financially supported by the National Natural Science Foundation of China (No. 81872775)。
The rapid prevalence of antibiotic resistance has led to a significant global health problem. Although colistin is the last resort antibiotic, it is limited by dose dependent toxicity. A critical approach to solve thi...
关键词：2-Aminothiazole piperidine Antibiotic adjuvant Acinetobacter baumannii COLISTIN 
Synthesis of 2-aminothiazoles via rhodium-catalyzed carbenoid insertion/annulation of sulfoxonium ylides with thioureas被引量：1
《Chinese Chemical Letters》2021年第8期2555-2558,共4页Yuncan Chen Shan Lv Ruizhi Lai Yingying Xu Xin Huang Jianglian Li Guanghui Lv Yong Wu 
support from the National Natural Science Foundation of China (Nos.81373259 and 81573286);Sichuan Science and Technology Program (Nos.2020YJ0221 and 2018JY0537)。
Sulfoxonium ylides as carbene precursors couple smoothly with thioureas in the presence of 5 mol% of rhodium(Ⅱ) acetate dimmer via carbenoid insertion to afford the corresponding 2-aminothiazoles with high chemoselec...
关键词：2-Aminothiazoles Carbene Rhodium Sulfoxonium ylides ANNULATION 
Synthesis, Antitumor Activity and Preliminary Structure-activity Relationship of 2-Aminothiazole Derivatives被引量：3
《Chemical Research in Chinese Universities》2016年第6期929-937,共9页LI Hongshuang WANG Xinran DUAN Guiyun XIA Chengcai XIAO Yuliang LI Furong GE Yanqing YOU Guirong HAN Junfen FU Xiaopan 
In this paper, we described the synthesis of 2-aminoflfiazole sublibrary containing methyl, bromo, phenylor butylidene at 4- or/and 5-position of its core. All target compounds were evaluated tbr their antitumor activ...
关键词：2-Aminotlfiazole ANTITUMOR activity STRUCTURE-ACTIVITY RELATIONSHIP 
Discovery of novel dual inhibitors of VEGFR and PI3K kinases containing 2-ureidothiazole scaffold被引量：1
《Chinese Chemical Letters》2016年第1期1-6,共6页Lin Li Cun-Long Zhang Hong-Rui Song Chun-Yan Tan Huai-Wei Ding Yu-Yang Jiang 
the financial supports from the NSFC (No. 21272134);Shenzhen Municipal government SZSITIC (Nos. JCYJ20130402145002384, ZDSY20120619141412872)
A series of compounds possessing 2-（3-phenyl）ureidothiazol-4-formamide derivatives with a 2-ureidothiazole scaffold were designed and synthesized. Some compounds demonstrated inhibition of cell proliferation against...
关键词：2-AMINOTHIAZOLE VEGFR PI3 KAnticancer 
Synthesis and Antitumor Activity of 4-tert-Butyl-5-benzyl-2-benzyliminothiazoles被引量：1
《Chemical Research in Chinese Universities》2014年第1期49-54,共6页YE Jiao QIU Shenyi HU Aixi PENG Junmei QIN Zhi 
Supported by the National Science ＆ Technology Pillar Program of China（No.2011BAE06B01） and the Natural Science Foundation of Hunan Province, China（No. 12j j3012）.
A series of novel Schiff bases including 4-tert-butyl-5-benzyl-2-benzyliminothiazoles was synthesized by reacting the aromatic aldehydes with the corresponding 2-aminothiazoles.The antitumor bioassay revealed that com...
关键词：2-AMINOTHIAZOLE Schiff base Antitumor activity 
Polyfluoroalkylation of 2-Aminothiazoles： Unexpected sp3 C CI Substitution under Mild Conditions被引量：1
《Chinese Journal of Chemistry》2011年第12期2681-2683,共3页齐卿卿 沈其龙 吕龙 
Project supported by special Fund for Agro-scientific Research in the Public Interest （No. 201103007）, the National Key Technologies R＆D Program （No. 2011BAE06B05）, National Basic Research Program of China （No. 2010CB126103）, the Key Program of National Natural Science Foundation of China （No. 21032006） and SIOC startup fund.
An efficient, highly selective method for polyfluoroalkylation of 2-aminothiazole derivatives was described. Specifically, a di-polyfluoroalkylated derivative was produced when 2-amino-4-chloromethylthiazole was react...
关键词：POLYFLUOROALKYLATION 2-AMINOTHIAZOLE dipolyfluoroalkylation SULFINATODEHALOGENATION 
Synthesis and Biological Study of Some 4-oxo-Thiazolidine Derivatives of 2-Aminothiazole
《Chinese Journal of Chemistry》2011年第5期1001-1010,共10页Samadhiya Pushkal Sharma Ritu Srivastava Santosh K. Srivastava Savitri D. 
Conventional and microwave assisted synthesis of new series of N-[2-{2-（substituted phenyl）-4-oxo- 5-（substituted benzylidene）-1,3-thiazolidine}-iminoethyl]-2-aminothiazole 5a-Sin have been developed. The cycloadd...
关键词：conventional microwave SYNTHESIS 2-AMINOTHIAZOLE 4-oxo-thiazolidine ANTIMICROBIAL ANTITUBERCULAR 
One-pot synthesis of 2-aminothiazoles in PEG-400被引量：8
《Chinese Chemical Letters》2010年第4期412-416,共5页Dhanaji V.Jawale Dinesh L.Lingampalle Umesh R.Pratap Ramrao A.Mane 
A facile one-pot synthesis of 2-aminothiazoles has been carried in PEG-400 as a greener medium at room temperature.This method avoids the use of lachrymatric a-bromoketones as well as the volatile,toxic organic solvents.
关键词：One-pot synthesis 2-Aminothiazoles Polyethylene glycol-400 N-BROMOSUCCINIMIDE 
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