the Fundamental Research Funds for the Central Universities(22qntd2306);Guangzhou Municipal Science and Technology Bureau(202201011151);the National Natural Science Foundation of China(22201311).
Aromatic oxazolines are versatile in organic synthesis as directing groups,ligands,and protected carboxylic acids.Developing efficient approaches to oxazoline from an aromatic C−H bond is more desirable compared to th...
supported by the National Natural Science Foundation of China (No. 22078299);Zhejiang Provincial Natural Science Foundation of China (Nos. LY21B060005, LQ20B060007);the College of Pharmaceutical Sciences, Zhejiang University of Technology;Collaborative Innovation Center of Yangtze River Delta Region Green Pharmaceuticals for the financial help。
An efficient photocatalytic alkylation/cyclization of allylic amide with N-hydroxyphthalimide ester has been developed. The transformation is taken advantage of alkyl radicals to attack allylic amide with the assist o...
We appreciate the National Natural Science Foundation of China(21890723 and 21921002)for financial support.
An asymmetric Heine reaction of (meso)-N-(2-picolinoyl)-aziridines catalyzed by a chiral ytterbium(III)–N,N′-dioxide complex was established. A novel library of pyridine-oxazolines was obtained with decent yields an...
supported by the NSF of China(21572072);Xiamen Southern Oceanographic Center(15PYY052SF01);111 Project(BC2018061).
Photoredox-catalyzed generation of sulfonated oxazolines starting from N-allylamides,DABCO·(SO2)2,and aryldiazonium salts has been developed.A range of sulfonated oxazolines were obtained in moderate to good yields.T...
supported by the National Natural Science Foundation of China(Nos.21963008 and 21767010);the Natural Science Foundation of Hubei Province(No.2018CFB650);the Postgraduate Research and Innovation Plan Project of Hubei Minzu University(No.MYK2020001)。
Excited-state intramolecular proton transfer(ESIPT) reactions of three ortho-hydroxylated oxazolines, 2-(4,4-dimethyl-4,5-dihydro-oxazol-2-yl)-phenol(DDOP), 4-(4,4-dimethyl-4,5-dihydro-oxazol-2-yl)-[1,1?-biphenyl]-3-o...
the National Natural Science Foundation of China(No.21702106);the Natural Science Foundation of Jiangsu Province(No.BK20170967);the Start-up Grant from Nanjing Tech University(No.39839101)for financial support。
Disclosed herein is an efficient Ag-catalyzed 4+1 heteroannulation reaction of enamides withα-carbonyl sulfoxonium ylides.The diastereoselective transformation provides a practical access to a diverse range of multi-...
partial financial support from the Ministry of Science and Technology of China(No.2016YFE0132600);Zhengzhou University。
A selective ring-opening [3+2] cyclization reaction of benzo[d]isoxazoles with 2-bromo-propanamides has been developed.The azaoxyallyl cation intermediates are employed as C^O 3-atom synthon to build oxa-heterocycles ...
Supported by the National Natural Science Foundation of China(Nos.20572066, 20906059) and the Natural Science Founda- tion of Shaanxi Province of China(No .2009JM2011).
An efficient method for the one-pot synthesis of 2-oxazolines from ethyl a-cyanocinnamate derivatives with acetamide and N-bromosuccinimide(NBS) in the presence of K3PO4 was developed. The reaction was performed smo...
Project supported by National Natural Science Foundation of China (No. 20672016).
2-Oxazolines and 2-benoxazoles were synthesized in high yields from acylamino alcohols and acylaminophenols, respectively, with triphenylphosphine-2,3-dichloro-5,6-dicyanobenzoquinone (PPh3-DDQ) as the dehydrating a...
Chloroamidinium salts and a-amino alcohols derived from commercially available tetraalkyl ureas and α-amino acids, respectively, can be used for the syntheses of optically active 2-(N,N-dialkylamino)oxazolines in m...